Izidakamizwa ezingavimba ukuvuvukala emakethe yanamuhla yezokwelapha zihanjiswa ngezindlela ezihlukahlukene - kokubili ngamapulders, nasezibhebheni, nasezijoweni, futhi-ke, ngendlela yamafutha namafutha. Enye ye-NSAID ethandwa kakhulu ngesimo se-gel ingabizwa nge-Diclofenac. Lokhu kungenxa yezici eziningana: okokuqala, lesi sidakamizwa asinayo intengo ephakeme, futhi okwesibili, sisebenza kahle, futhi, okwesithathu, ukuthandwa kwegama lomuthi kusekelwa ezinye izinhlobo - izijovo ezifanayo namaphilisi.
Ukwakhiwa kwe-gel Diclofenac
I-Diclofenac imelela ama-anti-inflammatory non-steroid agents futhi iqukethe i-gel kusuka e-diclofenac sodium.
Izinto ezisizayo ezisiza i-gel ukuba ingene kahle zibe izicubu futhi zigcine izindawo zayo isikhathi eside ziyizi:
- i-ethanol ilungiswe;
- i-propylene glycol;
- i-triethanolamine;
- i-carbomer;
- i-methyl lauryl hydroxybenzonate;
- i-lavender amafutha;
- amanzi ahlanzekile.
Ukukhululwa kwefomu nokuxilongwa kwe-gel Diclofenac
I-Gel Diclofenac itholakala kuma-tubus aluminium ama-50 no-40 g.
Ngaphandle kwevolumu, ukuhlushwa kwezinto ezihlukile kubuye kuhluke:
- I-gel Diclofenac 5% - ngayinye yegremu eyi-1 g yenza ama-50 mg we-diclofenac sodium;
- I-gel Diclofenac 3% - 1 g yama-gel ama-30 mg we-diclofenac sodium;
- I-gel Diclofenac 1% - i-1 g yejel ayi-10 mg yesithako esikhulu esisebenzayo - i-diclofenac sodium.
Amafutha e-Diclofenac akakho, kuphela i-gel iyatholakala.
Izakhiwo zomzimba ze-gel Diclofenac
I-Diclofenac iyisisombululo esinomphumela we-analgesic, kanye nokubiza izakhiwo eziphikisayo. Ivimbela ama-enzymes COX-2 ne-COX-1, futhi iphazamisa ukuhlanganiswa kwe-arachidonic acid kanye nokusetshenziswa komzimba we-prostaglandins, okwenza uchungechunge lokuvuvukala. Ngakho, i-gel igqugquzela ukusabalala kokuvuvukala, futhi ivimbela ukuthuthukiswa kwayo ezakhiweni ezizungezile.
Ngenxa yalezi zakhiwo, i-Diclofenac isetshenziswa njenge-decongestant uma ukuvuvukala kubangelwa ukuvuvukala. Kubuye kunqunywe ukuhlukunyezwa kobuhlungu njenge-anesthetic yangakini uma ubuhlungu bubangelwa inqubo yokuvuvukala.
I-Diclofenac inciphisa ukuvuvukala ezindaweni zokuvuvukala okuhlangene, ukukhulula ukuqina. Kanti futhi ezindaweni zokuvuvukala, noma ukuqeda ubuhlungu, noma ngokunciphisa kakhulu.
Imiyalelo ye-gel Diclofenac
Imiyalo yokusetshenziswa kwe-Diclofenac Gel 5%, kanye no-3% no-1% ayifani. Umehluko ukhona ekugxilweni kwemithi esebenzayo, futhi inhloso yayo ixhomeke ebukhulu bezimpawu. Isibonelo, i-gel Diclofenac ene-concentration ye-5% isetshenziselwa ukuphatha ubuhlungu obukhulu e- rheumatism .
Izinkomba zokusebenzisa i-gel Diclofenac
I-Diclofenac inqunywe ngezifo ezilandelayo:
- pathologies rheumatic - bursitis , tendovaginitis, njll ;;
- Ubuhlungu be-muscle ngemuva kwe-rheumatism noma ukulimala kwezicubu zomzimba;
- ukuvuvukala kwe-posttraumatic kwamalungu.
Ijelisi le-Diclofenac lisetshenziswa ngaphandle, futhi inani lokusetshenziswa okulodwa lingcike ngobukhulu bendawo ebuhlungu.
Noma kunjalo, kunezincomo ezijwayelekile zokusetshenziswa kwe-gel yezingxube ezahlukene:
- I-gel Diclofenac 1% - ukusetshenziswa okukodwa - kufika ku-4 g;
- I-gel Diclofenac 3% - ukusetshenziswa okukodwa - kufika ku-3 g;
- I-gel Diclofenac 5% - ukusetshenziswa okulodwa kuze kube ngu-2 g.
Izingane ezineminyaka engaphezu kwengu-12 kanye nabantu abadala bakhuthazwa ukuba basebenzise i-gel 3-4 izikhathi ngosuku ngokunyakaza okukhanyayo.
Ukungafani kokusetshenziswa kwe-gel Diclofenac
I-Diclofenac ayikwazi ukusetshenziswa kulezi zimo ezilandelayo:
- ukukhulelwa (isincomo 3 trimester);
- i-lactation;
- iminyaka yezingane (kuze kube yiminyaka engu-6);
- amanxeba, ukushisa;
- ukusabela okweqile noma i-asthma ebangelwa ukusetshenziswa kwezidakamizwa ezingezona ukuvuvukala.
Uma kunesifo sokuphuma kwegazi, i-Diclofenac Gel 5% kufanele isetshenziswe ngokucophelela.