I-Desloratadine ne-loratadine - umehluko

Ukuze uqonde ngokushesha ukuthi yini i-desloratadine, khumbula isidakamizwa esidumile njengo- Erius . Lesi yisisombululo esivamile kakhulu sokwelapha izifo. Isithako sayo esisebenzayo, i-desloratadine, iyisimetabolite ye-loratadine. Lesi sici senze imiphumela ehlukile yezinto ezimbili. I-Desloratadine ne-loratadine, umahluko ophikisiwe ngezansi, ngokuphumelelayo ukulwa nokuxoshwa kwezinto ezihlukahlukeneyo, ukukhulula ukukhukhumeza nokusebenzisa isenzo sokuphikisa.

Uyini umehluko phakathi kwe-loratadine ne-desloratadine?

Zombili izinto zivimbela i-histamine n1 receptors. Abanayo isenzo se-cardiotoxic ne-hypnotic, basuswa ngokushesha emzimbeni ngaphandle kokulibala.

Nokho, i-desloratadine iyi-metabolite ye-loratadine, okungukuthi, umkhiqizo wokucubungula. Ngakho-ke, lapho ethatha i-loratadine, yena, ngaphambi kokuqala isenzo sakhe, uphenduka i-desloratadine. Ngakho-ke, lesi samuva siqala ngokushesha kakhulu kunokulungiswa kwesizukulwane esedlule, ngoba akudingeki siguqulwe sibe yimpahla yokugcina.

Yikuphi okungcono - i-desloratadine noma i-loratadine?

Izinzuzo ze-desloratadine zihlanganisa ukusebenza kahle kwazo. Kuyizikhathi eziphindwe izikhathi ezingu-4-15 ezisebenzayo kunokuba zilandelwe ngaphambili. Lokhu kuvumela ngokushesha ufinyelele ukuhlushwa okuphezulu futhi unciphise umthamo ngesigamu.

Kufanele kuqaphele ukuthi izidakamizwa eziningi ezisuselwa ku-desloratadine zithengiswa njenge-siraphu, okwenza kube lula ukuphatha izingane, kuqala ngezinyanga eziyisithupha.

Ukucubungula i-desloratadine kanye ne-loratadine bese uphendula lo mbuzo ukuthi umehluko ophikisayo, kufanele kuqaphele ukuthi uma lokhu okudingekayo kudingeke, ukusebenza okujwayelekile kwesibindi kuyadingeka. Phela, uma kwenzeka noma yikuphi ukugula, ukuguqulwa kwe-desloratadine ngeke kwenzeke.

Izindleko zezidakamizwa ezisekelwe ku-desloratadine yi-oda lobukhulu obuphakeme kunele-loratadine. Imithi yokugcina kufanele inikezwe uma kunesidingo ukulwa nezimo ezilodwa zokungezwani komzimba , ngokungabikho kwezifo zesibindi.