I-Diclofenac yiqembu lemithi esetshenziselwa izifo ezihlukahlukene zokuvuvukala kwamalungu kanye nemisipha. Into esebenzayo yalesi sidakamizwa ibhekisela emithini engeyona-steroidal elwa nokuvuvukala, eneziningi zokuphikisana nemiphumela emibi. Kule ndaba, kuvame ukuba nesidingo sokuthola i-analog - ephumelela ngokwengeziwe futhi ngesikhathi esifanayo. Futhi, akekho kodwa ukhombise ukuthi ososayensi base-UK bacela ukususwa kukaDiclofenac ngoba, ngokuhambisana nezifundo zabo, kwandisa kakhulu ingozi yokuhlaselwa yinhliziyo , okuyiyona namuhla "yezingxabano" eziyinhloko zesintu. Le kholi yayingathinti kakhulu odokotela basekhaya, kanti uDiclofenac usalokhu enqunywe ukuba athole ukwelashwa.
Okulandelayo, sizobuka imithi engayenza esikhundleni seDiclofenac.
Ama-analogs e-Diclofenac ku-Injections kanye nolwazi olujwayelekile
Ama-analogues e-diclofenac emajenjini awanzima ukuthola, uma ubheka isimiso somuthi osebenzayo ofanayo. I-diclofenac sodium iqukethwe kuVoltaren, Diklak, Almiral, nabanye.
Kunzima kakhulu ukuthola i-ejenti efanayo nomunye umsebenzi osebenzayo. Uyi-Arthrosan - into eyinhloko esebenzayo - i-meloxicam. I-inhibitor ekhethiwe ye-COX-2, futhi futhi emele izidakamizwa ezingezona ukuvuvukala okungezona ama-steroidal, nge-biovailability enkulu ye-89%. Kuyathakazelisa ukuthi i-Diclofenac, ngokusho kwemiyalo, ivumelekile ukuthi isetshenziswe ngesikhathi sokukhulelwa, uma ukusetshenziswa kwayo kuzibeka eqondile ngenxa yobungozi kwengane nomama, futhi, ngesikhathi esifanayo, i-Arthrosan iphikisana ngokuphelele ekukhutheni.
Ngakho-ke, kungashiwo ukuthi i-Diclofenac iyisiluleko samanje nesiphephile, naphezu kwesixwayiso ososayensi baseBrithani. I-arthrosan inemiphumela eminingi emibi evela kuzo zonke izinhlelo zomzimba.
I-Analog Diclofenac e-ampoules ngendlela ye-meloxicam akufanele isetshenziswe isikhathi eside.
I-analogue yesimanje yeDiclofenac yiNaproxen. Ihlinzekwa ngesimo sejoza, ama-gel kanye namathebulethi, inomthelela obuthakathaka kune-sodium diclofenac, kodwa ngesikhathi esifanayo yisidakamizwa esinamandla.
I-Naproxen ibhekisela ngesikhathi esisodwa kumaqembu ama-pharmacy amahlanu:
- i-spasmoanalgesic;
- Ama-NSAID ahlanganisiwe;
- i-analgesic-antipyretic enezinto ezihlanganisiwe;
- Ama-NSAID ahlanganiswe neproton pump inhibitor;
- Ama-NSAID.
Esinye isidakamizwa esivimba ukuvuvukala esingashintsha i-Diclofenac ngu-Ibuprofen. Eqinisweni, lokhu kuyi-analog yayo uma siqhathanisa nemiphumela emibi, izinkombandlela kanye nezinkomba. U-Ibuprofen ungumphumela we-phenylpropionic acid, futhi, njengamanye ama-NSAID, avimbela i-COX.
Ama-analogues e-Diclofenac kumathebulethi
Ama-analogs e-Diclofenac kumaphilisi, ngaphezu kwezimali ezingenhla, yi:
- I-Clofezon;
- Sulindak;
- Indomethacin;
- I-Piroxicam;
- I-Tenoxicam.
Kumele kuqashelwe ukuthi uSulindack akayona ingozi kakhulu kwesisu kune-Indomethacin, kodwa ngesikhathi esifanayo isifo esinobuthi kakhulu esibindi.
Ama-analogues e-diclofenac ointment
- Ketoprofen;
- I-Phenylbutazone (i-Butadione);
- I-Clofezon;
- Indomethacin.
Amafutha amaningi aphephile phakathi kwama-Doglofenac i-Clofezon. I-Phenylbutazone ibekezelela kakhulu, kepha idlula i-aspirin ngomphumela wayo. I-Indomethacin yisidakamizwa esinamandla kunazo zonke esingazange steroidal anti-inflammatory, ngakho-ke sinqunywe ezimweni ezimbi kakhulu, ngenkathi kubangela umonakalo omkhulu emzimbeni.
Ama-analogue e-Diclofenac
- I-Naproxen;
- Ketoprofen;
- Ukuphakama;
- Piroxicam.
Izakhiwo ezinamandla kunazo zonke phakathi kwama-gel yiPiroxicam noKetoprofen. I-naproxen evame ukusetshenziswa kakhulu ingenxa yokubuthakathaka
Analogues of amakhandlela Diclofenac
- I-Metamizole;
- Fenacetin;
- I-Clofezon;
- Indomethacin;
- I-Naproxen;
- I-Tenoxicam.
I-Indomethacin yimithi ephumelela kakhulu yaleli qembu, ngakho-ke akukhuthazwa ukuyisebenzisa njalo.