Josamycin analogues

I-Josamycin kanye nezifanekiselo zalo ziyingxenye yeqembu elimangalisayo. Lezi zidakamizwa zinomthelela we-bactericidal. Into esebenzayo ixhumana ne-sub-50S, ivikela ukugcinwa kwe-RNA yezokuthutha kanye nokucindezela amaprotheni synthesis.

Yini engayenza esikhundleni sikaJosamycin?

Imithi iboniswa ngezifo ezingapheli futhi ezinzima ezibangelwa ukuphazamiseka kwe-microflora. Ukuze ubuyisele umsebenzi ovamile, ngokuvamile usebenzise izidakamizwa ezisekelwe ku-josamycin. Ngokuvamile le mithi enegama elifanayo. Unomthelela othize emzimbeni, ususe izimpawu eziningi. Nanobe kunjalo izifanekiselo ezivamile nezindlela ezishibhile zikaJosamycin.

Isibonelo, okuvame kakhulu kubhekwa ukuthi nguWilprafen. Lena iphilisi. Kuboniswa ukwelashwa:

Ngaphezu kwalokho, i-generamic ejwayelekile kaJosamycin ibhekwa njengeVilprafen solute. Lesi sidakamizwa i-analog ephelele. Ibuye inezindawo zokulwa ne-antibacterial and bactericidal. Kodwa nokho kukhona umehluko - amaphilisi anikezwa ifomu elingu-oblong, ayamnandi futhi anelungelo lokunuka kwe-strawberry.

Izilinganiso zalesi sidakamizwa nazo zibhekwa njengama-antibiotics weqembu le-macrolide:

Uhlobo luni lomuthi olulungele lokhu noma lesi siguli, kuzoba ochwepheshe kuphela abazokwazi ukuthola, ngokusekelwe ezinkomba zokuhlaziya. Ngokuvamile ungakuzwa ukuthi uma kungekho muthi ekhemisi, khona-ke ushintshwe ngokuphepha ngomunye. Kodwa lokhu akulona iqiniso elingu-100%. Esikhathini ngasinye, ukubonisana nodokotela kuyadingeka.

Yini engcono - i-Jozamycin noma i-Azithromycin?

Abaningi babanika lezi zidakamizwa, ngaphandle kokungabaza: basebenzisa cishe into esebenzayo, ngakho-ke umphumela wabo okufanayo. Naphezu kwalokhu, ngokusekelwe ezifundweni zamazwe ngamazwe, singasho ngokuphepha ukuthi i- Azithromycin iholela kancane ekubonisweni kwemiphumela emibi njengo: