Ama-analogues e-Roxer

Izidakamizwa ze-gipolipidemic zibalulekile kulabo bantu abadinga ukuhlola njalo izinga le- cholesterol egazini. Ukulungiswa kwe-Roxer nama-analogs alo kudalwe ngokukhethekile kule njongo. Ukulawula inani le-cholesterol emzimbeni kuzosiza ukuvimbela inani elikhulu lezifo futhi kuzoqinisekisa impilo enhle.

Izinkomba zokusetshenziswa kwezidakamizwa i-Roxer nezifanekiselo zayo

Into esemqoka yokusebenza kwe-roxera i-rosuvastine. Kuyinto inhibitor ye-enzyme ekhethekile - i-HMG-CoA iyanciphisa, - iyingxenye yokwakheka kwe-cholesterol. Ngaphandle kwe-rosuvastine, i-Roxer ihlanganisa izingxenye ezinjalo ezisizayo njenge:

Kokubili imithi yama-Roxer kanye ne-analog isenza esibindi - esithombeni lapho i-cholesterol iklanyelwe khona. Izidakamizwa zithuthukisa ngokuphumelelayo inani le-receptors ye-hepatic, ngaleyo ndlela kuncishisa izinga le-lipoprotein cholesterol elincane.

Izidakamizwa ezikhethiwe zezilwane ezinjalo:

Yini engcono - i-Roxer, i-Atoris noma i-Krestor?

Naphezu kokuthi i-Roxera ibhekwa njengomuthi osebenzayo futhi ophephile, ngesizathu esithile umuthi awufanele wonke umuntu. Iziguli ezinjalo zidinga imithi efanayo. I-Atoris ne-Krestor baba yizifaniso ezidume kakhulu ze-Rockers. Isimiso sokusebenza salezi zidakamizwa cishe sifana. Umehluko oyinhloko usekubunjweni.

Into esemqoka esebenzayo eRoxer naseKrestor yi-rosuvastine. Okusho ukuthi, lezi zidakamizwa cishe zifana. Ahluke kumkhiqizi, ngakho-ke, futhi ngentengo - i-Crestor iyabiza kakhulu. Ezinye iziguli ziphawula ukuthi iKrestor yenza ngokushesha, kodwa lokhu kuncike kakhulu ekuziphatheni komzimba, ubuciko, ukuxilongwa.

Njengengxenye yesinye isifaniso se-Roxer - amaphilisi e-Atoris - atorvastatin. I-Atoris cishe isilinganiso samanani afana ne-Roxer, kodwa ihamba kancane, ngakho odokotela bakhetha ukuyibeka njengesilinganiso sokuvimbela nokwelapha izifo ezisezigaba zokuqala.

Ngokwenzayo, kuyindlela kuphela yokuhlola esiza ukunquma ukuthi iyiphi imithi esebenza kangcono kwelinye icala noma kwelinye icala. Ngokuvamile kwenzeka ukuthi ezinye izidakamizwa zilungele omunye umuntu, kodwa kumuntu ongenzi lutho ngokugcwele.

Ungayinqoba kanjani i-Roxer?

Yiqiniso, ngaphezu kwamalungiselelo e-Atoris naseKrestor, kunezinye izizukulwane zikaRoxer. Ngaphezu kwalokho, uhlu lwabo luyamangalisa:

Umphumela wokuthatha ama-statins ufika emavikini ambalwa emva kokuqala kokwelashwa. Isilinganiso nesikhathi sokuthola ukwelashwa ngoba isiguli ngasinye sinqunywe ngabanye.

Futhi ukulungiswa kweRoxer, futhi okufana nezigaba ezithile zeziguli kuyaphikisana:

  1. Ungathathi ama-statins omama abakhulelwe nabaqabulayo.
  2. Ukwelashwa ne-Roxer kanye nezifanekiselo zalo kuphikisana nabantwana abangaphansi kweminyaka engu-18 ubudala.
  3. Ungafanisi izidakamizwa ze-statin kubantu abanezinso ze-kidney.
  4. Ukulimaza i-Roxer kanye nama-analogs ayo kungaba neziguli ezinezifo ze-neuromuscular.