Ama-analogue e-Verapamil

I-Verapamil yisidakamizwa esithengiswa ngesimo samathebulethi agcwele i-film coating noma ngendlela yethebhulethi enesisindo esingama-40 noma i-80 g. Isenzo eside se-Verapamil sithengiswa ngephakhethi ebizwa nge-Verapamil 240, futhi, njengokubusa, izifanekiselo zalo zinesenzo esifanayo. Imithi enjalo inqunywe ngendlela yamajojo nge:

Yini engayenza esikhundleni se-verapamil?

Kunezifanekiselo ezimbalwa ze-Verapamil yezidakamizwa. Zonke zifana nokusebenza okusebenzayo okukhulu - i-verapamil futhi kuboniswa:

Nalu uhlu lwemithi ejwayelekile kakhulu engasetshenziswa esikhundleni se-verapamil:

Ukusetshenziswa kwezidakamizwa ze-Verapamil nama-Analogue awo

I-Verapamil ekubunjweni kwawo wonke amalungiselelo afanayo alungiswayo enza ukuba ukwandiswa kwemithambo ye-coronary kanye ne-arterioles ejwayelekile kanye nezindawo zenhliziyo, lapho igazi linciphisa khona ngenxa yokunciphisa umzimba. Isenzo sezidakamizwa sivimbela ukugawula izikebhe ze-coronary, ngaleyo ndlela kuthuthukise ukunikezwa kwegazi emisipha yenhliziyo.

I-Verapamil nama-analogs awo awavumeli ion calcium ukuba idlule emangqamuzaneni eseli, okuholela ekunciphiseni izinga lokushaya kwenhliziyo nokunciphisa ukuphikiswa komuntu ngamunye kwemikhumbi. Ngakho-ke, umthwalo osiswini somzimba uyanciphisa kakhulu futhi igazi lalo landa. Into esebenzayo I-verapamil inciphisa isidingo se-myocardial emoyeni.

Kufanele ngithathe kanjani i-Verapamil nezithombe zayo ezifanayo?

Amathebulethi i-Verapamil kanye nezifanekiselo zalo kuthathwa ngesikhathi sokudla noma ngokushesha emva kokudla, ngaphandle kokuhlafuna ukugwinya nokugeza ngamanzi.

Ngaphambi kokusebenzisa izidakamizwa, kudingeka uqiniseke ukuthi azikho izifo ezithintekayo, ngoba uhlu lwezinqununu lukhulu kakhulu. Akunconywa ukuthi uthathe i-Verapamil nezidakamizwa ezifanayo ngesikhathi sokukhulelwa kanye ne-lactation.