I-Diphenin analogues

Isidakamizwa se-Anticonvulsant i-Diphenin sinemifanekiselo, lapho ekubunjweni kwayo nokusebenza kwayo akuzona ngaphansi kwale mithi.

Izici zesidakamizwa i-Diphenin kanye nezifanekiselo zayo

Isidakamizwa singumuthi we-hydantoin. Inomphumela olandelayo:

Ngesikhathi sokudliwa kwamaphilisi e-Diphenin, kutholakala kancane kancane. I-Phenitonin, engxenyeni yesidakamizwa, ifinyelela ebuchosheni bobuchopho, emathunjini, esiswini, nangomusi wamathumbu. Kungabuye kukhishwe ngobisi lwebele, okwenza kube yingozi kumntwana futhi kuvinjelwe ngesikhathi sokulahlwa. Kulesi simo, isidakamizwa senziwa ngokweqile ngokusebenzisa izinso ngendlela yama-metabolites, bese-ngaphakathi kwamathumbu.

Njenganoma imuphi umuthi, i-Diphenin inezinamba eziningi zokuphikisa:

Kumele kuthiwa izidakamizwa nezidakamizwa ezifanayo zinemiyalelo ekhethekile ngesikhathi sokusebenza. Isibonelo:

  1. Kubalulekile ukuhlola njalo ukuhlushwa kwe-phosphorus ne-calcium e-serum yegazi.
  2. Abantu abanesifo sokuphuza kufanele kancane kancane bayeke umuthi noma bashintshele kwenye i-anticonvulsant ngaphandle kokutholakala kwe-hydantoin, njengoba ukuguqulwa okungazelelwe kungaholela emiphumeleni emibi.
  3. Ungahlanganisi i-diphenin ne-acetazolamide, ngoba kungase kube khona ingozi yokuthuthukisa ama-rickets noma i-osteomalacia.
  4. Ukuhlanganisa umuthi onjalo neGabalentin kungabangela ukuthuthukiswa kwemiphumela enobuthi.
  5. Amathebulethi aqukethe i-phenytoin, avimbela ukusabela kwengqondo, ngakho-ke abantu abahlale beqaphele futhi basabela ngokushesha kulokho okwenzekayo, le mithi iphikisana.

Ungashintsha kanjani i-Diphenin?

Labo abanesithakazelo kulo mbuzo, yini engayenza esikhundleni seDifenin, kufanele ubone uhlu olungezansi. Ibala imishanguzo efana nezinkomba zokusetshenziswa nokusebenza kwemithi. Imithi elandelayo ifana nalokhu: